Ярославль, Ярославская область, Россия
Ярославль, Ярославская область, Россия
Ярославль, Ярославская область, Россия
Ярославль, Ярославская область, Россия
УДК 547-304.7 Нитрилы. Изонитрилы
The paper presents a preparation method for 3-cyanobenzene-1-sulfonyl chlorides, valuable reagents for the fine organic synthesis used in the preparation of antiplatelet agents and agricultural germicides, pharmaceutical compositions, and biologically active compounds.
preparation method, 3-cyanobenzene-1-sulfonyl chlorides, antiplatelet agents, agricultural germicides
1. Perzborn E., Seuter F., Fruchtmann R., Kohlsdorfer C. Substituted phenyl-sulphon amides. Patent No. DE3632329(A1) Germany. No. 19863632329, publ. 31.03.1988.
2. Igarashi K., Enomoto Y., Yanagida H., Gohara M., Iida N., Ozawa S., Kuwazuka T. Sulfonamide based compound and agricultural germicide. Patent No. JPH0655708 (B2) Japan. No. 19850099595, publ. 27.07.1994.
3. Witte E.-C., Stegmeier K., Doerge L. Sulfonamidoalkyl cycloalkane compounds, processes for their production and pharmaceutical preparations. Patent No. DE3829455(A1) Germany. No. 19883829455, publ. 15.03.1990.
4. Witte E.-C., Stegmeier K., Dorge L., Doerge, L. Sulfonamidoalkyl cycloalkane compounds, processes for their production and pharmaceutical preparations. Patent No. EP0361113 (B1) Europe. No. 19890115912, publ. 07.07.1993.
5. Owa T., Yoshino H., Okauchi T., et al. J. Med. Chem. 1999. V. 42. N. 19. P. 3789-3799.
6. Wakabayashi T., Ono N., Semba T., Haneda T. Antitumor agent comprising combination of sulfonamide-containing heterocyclic compound with an angiogenesis inhibitor. Patent No. US2005119303 (A1) USA. No. 20040504676, publ. 02.06.2005.
7. Mrozik H. Anthelmintic substituted sulfonamide derivatives: Application US3953492 (A) USA. No. 19750562712, publ. 27.04.1976.
8. Hagmann W., Lin L., Liu P., Mumford R., Reger T., Smith N., Stock N., Zunic J. Vla-4 antagonists. Patent No. US2007179190 (A1) USA. No. 20050591820, publ. 02.08.2007.
9. Reger T.S., Zunic J., Stock N., et al. Bioorg. Med. Chem. Lett. 2010. V. 20. N. 3. P. 1173–1176.
10. Aldrich Chemistry 2012-2014: Handbook of Fine Chemicals. Sigma-Aldrich, 2011. P. 3216.
11. Gilbert E.E. Sulfonation and related reactions. New York: Interscience Publishers, 1965. 529 p.
12. Cremlyn R.J. Chlorosulfonic acid: A versatile reagent. RSC Publishing, 2002. 322 p.
13. Malet-Sanz L., Madrzak J., Ley S.V. Preparation of arylsulfonyl chlorides by chlorosulfonylation of in situ generated diazonium salts using a continuous flow reactor. Org. Biomol. Chem. 2010. N. 8. P. 5324-5332.
14. Tarasov A.V., Moskvichev Ju.A., Pisarev P.K., Nikiforova A.A. Method for preparing arylchlorosulfonyl benzamides from benzoic acids. Invention Patent No. RU2298548C1, 10.05.2007.
15. Comprehensive organic chemistry: The synthesis and reactions of organic compounds. A series of 6 volumes. Edited by D. Barton and W.D. Ollis. Volume 2. Nitrogen Compounds. Pergamon Press. 1979.
16. Harrison I.T., Harrison S. Compendium of organic synthetic methods. John Wiley & Sons, Inc. 1971. 529 p.
